Tag: Cholinergic Antagonist
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Belladonna alkaloids/Phenobarbital
Brands Classes DEA Class; Rx Common Brand Names; Donnaphen, Donnatal, Donnatal Extentabs, Haponal, Hypersed, Phenohytro, Spacol Belladonna (incl derivatives) and Psycholeptic Combinations atropine sulfate/hyoscyamine sulfate/phenobarbital/scopolamine hydrobromide Description Phenobarbital; hyoscyamine; atropine; scopolamine are used together orally to treat GI-related problems such as irritable bowel syndrome. Atropine, hyoscyamine, and scopolamine are the anticholinergic agents found in belladonna.…
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Terbutaline
Brands Classes DEA Class; Rx Common Brand Names; Brethaire, Brethine, Bricanyl Beta2 Agonists; Extravasation Antidotes Description Systemic short-acting selective beta-2 agonist (SABA); shorter acting than albuterolUsed for treating and preventing bronchospasm due to asthma in adult and pediatric patients; also for bronchospasm due to COPD in adults, but inhaled agents are preferredNot recommended for use…
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Vecuronium
Brands Classes DEA Class; Rx Common Brand Names; Norcuron Neuromuscular Blockers, Nondepolarizing Description Parenteral, intermediate-acting, nondepolarizing, neuromuscular blocking agentUsed for an adjunct to general anesthesia to facilitate endotracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilationMinimal catecholamine and histamine release Indications Indicated For muscular relaxation during non-emergent endotracheal intubation. For…
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Succinylcholine
Brands Classes DEA Class; Rx Common Brand Names; Anectine, suxamethonium, Quelicin Neuromuscular Blockers, Depolarizing Description Parenteral, short-acting, depolarizing neuromuscular blocking agent (NMBA)Used for an adjunct to general anesthesia to facilitate tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilationAssociated with histamine release and vagal stimulation Indications Indicated For muscular relaxation during…
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Rocuronium
Brands Classes DEA Class; Rx Common Brand Names; Zemuron Neuromuscular Blockers, Nondepolarizing Description Parenteral, intermediate-acting, nondepolarizing, neuromuscular blocking agent (NMBA)Used for an adjunct to general anesthesia to facilitate both rapid-sequence and routine tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilationMinimal histamine release Indications Indicated for muscular relaxation during non-emergent…
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Pancuronium
Brands Classes DEA Class; Rx Common Brand Names; Pavulon Neuromuscular Blockers, Nondepolarizing Description Parenteral, long-acting, nondepolarizing, neuromuscular blocking agentUsed for an adjunct to general anesthesia to facilitate tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilationMinimal histamine release; associated with tachycardia and hypertension due to vagolytic properties Indications Indicated for…
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Cisatracurium
Brands Classes DEA Class; Rx Common Brand Names; Nimbex Neuromuscular Blockers, Nondepolarizing Description Parenteral, intermediate-acting, nondepolarizing, neuromuscular blocking agent (NMBA)Used for an adjunct to general anesthesia to facilitate tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilationMinimal histamine release Indications Indicated for muscluar relaxation during non-emergent endotracheal intubation. For neuromuscular…
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Nicotine
Brands Classes DEA Class; Rx,OTC Common Brand Names; Nicorette Lozenge, Nicorette Mini Lozenge, Nicorette Inhaler, Nicotrol Inhaler, Nicotrol NS, Nicoderm CQ, Nicotrol, Nicorette Gum Smoking Cessation Aids Description Natural alkaloid of complex pharmacology inherent to the autonomic nervous systemUsed primarily for non-prescription (OTC) therapy to aide smoking cessation (patches, gum, lozenges); vaping solutions and…
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Trospium Chloride
Brands Classes DEA Class; Rx Common Brand Names; Sanctura, Sanctura XR Anticholinergics, Genitourinary Description Oral non-specific antimuscarinic agentUsed for the treatment of overactive bladder (OAB) in adultsDry mouth and constipation may occur; limited potential for drug-drug interactions Indications Indicated for the treatment of overactive bladder (OAB) with symptoms of urge urinary incontinence, urinary urgency,…
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Hydroxyamphetamine/Tropicamide
Brands Classes DEA Class; Rx Common Brand Names; Paremyd Cycloplegics/Mydriatics Description Topical ophthalmic combination of an adrenergic agent and an anticholinergic agentUsed for mydriasis in routine diagnostic procedures and in conditions where short-term pupil dilation desiredProvides diminished pupil responsiveness to light, facilitating ophthalmoscopy Indications Indicated for mydriasis induction in routine diagnostic procedures and conditions…
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Tropicamide
Brands Classes DEA Class; Rx Common Brand Names; Mydriacyl, Tropicacyl Cycloplegics/Mydriatics Description Ophthalmic cycloplegic and mydriatic agentUsed for cycloplegic refraction and for dilating the pupil for diagnostic purposesContraindicated for use in glaucoma Indications Indicated for cycloplegia induction for refraction. For mydriasis induction for examination of the fundus. Contraindications Hypersensitivity Known or suspected angle-closure glaucoma,…
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Trihexyphenidyl
Brands Classes DEA Class; Rx Common Brand Names; Artane, Trihex Antiparkinson Agents, Anticholinergics Description An oral synthetic, tertiary antimuscarinic that penetrates the central nervous system (CNS)Indicated as an adjunct in the treatment of all forms of parkinsonism (postencephalitic, arteriosclerotic, and idiopathic); often useful as adjuvant therapy with levodopaAlso helps control of extrapyramidal disorders due…
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Tolterodine
Brands Classes DEA Class; Rx Common Brand Names; Detrol, Detrol LA Anticholinergics, Genitourinary Description Oral competitive selective antimuscarinic agent; reduces incontinence episodes and urinary urgencyUsed for treatment of overactive bladder (OAB) in adults; used as monotherapy or in combination with a beta-3 adrenoreceptor agonist if neededExtensive study in elderly Indications Indicated for the treatment…
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Tiotropium/Olodaterol inhaled
Brands Classes DEA Class; Rx Common Brand Names; Stiolto Respimat Respiratory Inhalant Combos Description Inhaled long-acting muscarinic antagonist (LAMA), (tiotropium) with a long-acting beta-2 adrenergic agonist (LABA), (olodaterol); used once dailyUsed in adults for the maintenance treatment of COPD, including chronic bronchitis and/or emphysemaNot indicated for the relief of acute bronchospasm or for the…
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Tiotropium
Brands Classes DEA Class; Rx Common Brand Names; Spiriva HandiHaler, Spiriva Respimat Anticholinergics, Respiratory Description Inhaled long-acting muscarinic antagonist (LAMA); administered once daily; minimal side effects except for xerostomiaUsed for maintenance treatment of COPD in adultsAlso approved for maintenance treatment of asthma in adult and pediatric patients 6 years and older Indications For asthma…